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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 152368   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM152368
PNG
(US8993565, 97)
Show SMILES Cn1c(CC(=O)Nc2ccc(F)c(c2)C(F)F)nc(cc1=O)N1CCOCC1
Show InChI InChI=1S/C18H19F3N4O3/c1-24-14(23-15(10-17(24)27)25-4-6-28-7-5-25)9-16(26)22-11-2-3-13(19)12(8-11)18(20)21/h2-3,8,10,18H,4-7,9H2,1H3,(H,22,26)
PDB

UniProtKB/SwissProt
UniProtKB/TrEMBL

GoogleScholar
PC cid
PC sid
UniChem

Similars

US Patent
n/an/a 260n/an/an/an/an/an/a



Sanofi

US Patent


Assay Description
This test is based on measuring the expression of the AKT protein phosphorylated on serine 473 (P-AKT-S473), in the PC3 human prostate carcinoma line...


US Patent US8993565 (2015)


BindingDB Entry DOI: 10.7270/Q2FQ9V9P
More data for this
Ligand-Target Pair