TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 0.430nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 0.710nMAssay Description:Displacement of [125I]RTI-55 from recombinant human DAT expressed in CHOK1 cells after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina
Curated by ChEMBL
University Of North Carolina
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:The compound was tested for affinity towards sigma-3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of [125I]RTI-55 cocaine binding to the dopamine transporter.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Reuptake inhibition was determined at the dopamine transporter labeled with radioligand [3H]-dopamine in nonstandard conditions on brain membranes ob...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of dopamine transporter (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Dopamine uptake in male Sprague-Dawley rats using [3H]DA ligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Binding affinity was determined at the dopamine transporter labeled with radioligand [125 I] RTI-55 in nonstandard conditionsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of dopamine uptake at dopamine transporter.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Binding affinity was determined at the dopamine transporter labeled with radioligand [125 I] RTI-55More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Binding affinity for rat Dopamine transporter.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of [3H]GBR-12935 binding to the dopamine transporter.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Compound was tested for its ability to inhibit the uptake of [3H]-dopamine in DAT (dopamine transporter system) expressing cell lineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Compound was tested for its ability to inhibit the neurotransmitter dopamine-DA reuptake system using [3H]dopamine as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:The inhibition of reuptake of the compound against dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of dopamine DA reuptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Binding against Dopamine transporter using radioligand as [3H]GBR 12935More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 6.63nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Inhibition of human dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Reuptake inhibition at the dopamine transporter labeled with radioligand [3H]-dopamine on synaptosomes obtained from rat caudate.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Reuptake inhibition of [3H]-labeled dopamine (DA) in rat.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Inhibition of [3H]DA reuptake in rat caudate homogenate.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain homogenates after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:Inhibition of [3H]WIN-35428 binding to dopamine transporter of rat striatumMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:Binding affinity towards dopamine transporter in rat striatum using [3H]WIN-35 428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:Inhibition of binding of 3[H] WIN-35 428 to Dopamine transporter (DAT) of rat striatum.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:Binding affinity at the dopamine transporter in rast striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:Inhibition of [3H]-WIN- 35,428 binding to rat brain dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of binding of [3H]WIN-35 428 to (DAT) dopamine transporter in rat striatumMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]Win35428 from human recombinant DAT over-expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of [3H]-WIN- 35, 428 binding to dopamine transporter on rat striatal membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against dopamine transporter (DAT) labeled with [3H]-WIN- 35,428 in rat brain striatal membrane.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 14.2nMAssay Description:Inhibition of rat brain Dopamine transporter uptake as [3H]-DA accumulationMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 19.3nMAssay Description:IC50 value of the compound was evaluated using [3H]-WIN- 35,428 (radioligand) on Dopamine transporter in rat striatum.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 21.1nMAssay Description:Displacement of [3H]WIN 35428 from DAT in Sprague-Dawley rat striatumMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of [3H]BTCP binding to the dopamine transporter.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Affinity of the compound was evaluated using [3H]-DA (radioligand) on Cloned human Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of [3H]GBR-12935 binding to the dopamine transporter.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of [3H]cocaine binding to the dopamine transporter.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of re-uptake of [3H]-DA at human DAT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina
Curated by ChEMBL
University Of North Carolina
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Sigma receptor binding was determined by labeling with radioligand [3H]-(+)-pentazocine on frozen membranes obtained from frozen guinea pig brainMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Affinity of the compound was evaluated using [3H]-WIN- 35,428 (radioligand) on Cloned human Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of [3H]-5-dopamine reuptake in human DAT expressed in HEK293 cells by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Compound was tested for its ability to inhibit the neurotransmitter serotonin-5-HT reuptake system using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University Health Sciences
Curated by ChEMBL
Wake Forest University Health Sciences
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Reuptake inhibition at the dopamine transporter labeled with radioligand [3H]-5-HT on synaptosomes obtained from whole rat brain minus cerebellum.More data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Inhibition of [3H]5-HT reuptake at rat serotonin transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Inhibitory activity against [3H]- 5-hydroxytryptamine reuptake in whole rat brain minus cerebellumMore data for this Ligand-Target Pair