BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 292059   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Voltage-dependent calcium channel gamma-2 subunit


(Homo sapiens (Human))
BDBM292059
PNG
(2-(Difluoromethyl)-3-(7-methyl-1H-indazol-5-yl)-5-...)
Show SMILES Cc1cc(cc2cn[nH]c12)-c1n(nc2ccc(nc12)C(F)(F)F)C(F)F
Show InChI InChI=1S/C16H10F5N5/c1-7-4-8(5-9-6-22-24-12(7)9)14-13-10(25-26(14)15(17)18)2-3-11(23-13)16(19,20)21/h2-6,15H,1H3,(H,22,24)
PDB

UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
Article
US Patent
n/an/a 0.631n/an/an/an/a7.4n/a



Janssen Pharmaceutica NV

US Patent


Assay Description
Cell expressing the GRIA1o-CACNG8 fusion construct were grown in a monolayer in 96- or 384-well microtiter plates. They were washed with assay buffer...


US Patent US10100045 (2018)


Article DOI: 10.1021/jm049354h
BindingDB Entry DOI: 10.7270/Q2MW2K56
More data for this
Ligand-Target Pair