Affinity DataIC50: 290nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.25 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 20 uM) in OCT2-expressing HRPE cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Rattus norvegicus)
Medical College Of Georgia
Curated by ChEMBL
Medical College Of Georgia
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 20 uM) in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.07E+4nMAssay Description:TP_TRANSPORTER: inhibition pramipexole uptake in rOCT2-injected oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.17E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.25 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+4nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
Affinity DataIC50: 3.42E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.25 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.51E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.64E+5nMAssay Description:TP_TRANSPORTER: inhibition pramipexole uptake in rOCT1-injected oocytesMore data for this Ligand-Target Pair