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Found 5 of ic50 for monomerid = 50178612
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
The First People'S Hospital Of Hangzhou

Curated by ChEMBL
LigandPNGBDBM50178612((S)-4-((3-(dimethylamino)pyrrolidin-1-yl)methyl)-N...)
Affinity DataIC50:  4nMAssay Description:Inhibition of BCR-ABL kinase (unknown origin)More data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
The First People'S Hospital Of Hangzhou

Curated by ChEMBL
LigandPNGBDBM50178612((S)-4-((3-(dimethylamino)pyrrolidin-1-yl)methyl)-N...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of BCR-ABL (unknown origin) in presence of [gamma33P]-ATP and ATP by ELISA methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50178612((S)-4-((3-(dimethylamino)pyrrolidin-1-yl)methyl)-N...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human Lyn kinase expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50178612((S)-4-((3-(dimethylamino)pyrrolidin-1-yl)methyl)-N...)
Affinity DataIC50:  19nMAssay Description:Inhibition of LYN (unknown origin) in presence of [gamma33P]-ATP and ATP by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50178612((S)-4-((3-(dimethylamino)pyrrolidin-1-yl)methyl)-N...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human Abl kinase expressed in Sf9 cellsMore data for this Ligand-Target Pair