Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50299208
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50:  56nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50:  102nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1B receptor in Wistar rat liver membrane after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50:  320nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed