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Found 3 of ic50 for monomerid = 50303065
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50303065(3-(6-(4-chlorobenzylamino)pyrimidin-4-yl)pyrazolo[...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of JAK2 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50303065(3-(6-(4-chlorobenzylamino)pyrimidin-4-yl)pyrazolo[...)
Affinity DataIC50:  25nMAssay Description:Inhibition of JAK3 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50303065(3-(6-(4-chlorobenzylamino)pyrimidin-4-yl)pyrazolo[...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of JAK2-mediated STAT5 phosphorylation in GMCSF-stimulated human TF1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed