Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 50324430
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50324430((E)-3-(6-Methoxy-2-(4-nitrostyryl)-4-oxoquinazolin...)
Affinity DataIC50:  2.10E+4nMAssay Description:Antagonist activity at rat recombinant NR1-NR2C receptor expressed in Xenopus oocytes at holding potential of -40mV by two-electrode voltage-clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Emory University

Curated by ChEMBL
LigandPNGBDBM50324430((E)-3-(6-Methoxy-2-(4-nitrostyryl)-4-oxoquinazolin...)
Affinity DataIC50:  2.38E+5nMAssay Description:Antagonist activity at rat recombinant NR1-NR2A receptor expressed in Xenopus oocytes at holding potential of -40mV by two-electrode voltage-clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Emory University

Curated by ChEMBL
LigandPNGBDBM50324430((E)-3-(6-Methoxy-2-(4-nitrostyryl)-4-oxoquinazolin...)
Affinity DataIC50:  2.38E+5nMAssay Description:Antagonist activity at rat recombinant NR1-NR2B receptor expressed in Xenopus oocytes at holding potential of -40mV by two-electrode voltage-clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
Emory University

Curated by ChEMBL
LigandPNGBDBM50324430((E)-3-(6-Methoxy-2-(4-nitrostyryl)-4-oxoquinazolin...)
Affinity DataIC50: >3.00E+5nMAssay Description:Antagonist activity at rat recombinant GLuR1 expressed in Xenopus oocytes assessed as inhibition of glutamate-induced current by two-electrode voltag...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed