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Found 11 of ic50 for monomerid = 83205
TargetcAMP-dependent protein kinase catalytic subunit alpha(Rattus norvegicus (rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  98nMAssay Description:Inhibition of cAMP-dependent kinase PKA(Protein kinase A) catalytic subunit at 100 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-conjugating enzyme E2 N(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  6.20E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetUbiquitin-conjugating enzyme E2 N(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  6.43E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein kinase C zeta type(Rattus norvegicus)TBA
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibitory concentration required against Protein kinase C (isolated from rat brain) in PKC assay performed with 4 ug phosphatidyl serine:diacylglyce...More data for this Ligand-Target Pair
In DepthDetails
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  1.15E+4nMAssay Description:Compound was measured for its inhibitory activity against cholesteryl ester transfer protein (CETP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBcl-2-related protein A1(Mus musculus (Mouse))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50: >2.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetC-C chemokine receptor type 6(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  2.09E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego, CA...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein kinase C zeta type(Rattus norvegicus)TBA
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibition of Protein kinase C of rat brain using phosphatidyl serine: di-acyl glycerol (2:1)More data for this Ligand-Target Pair
In DepthDetails
TargetProtein kinase C zeta type(Rattus norvegicus)TBA
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibition of Protein kinase C isolated from rat brainMore data for this Ligand-Target Pair
In DepthDetails
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50:  5.70E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM83205((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...)
Affinity DataIC50: >6.66E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego, CA...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay