Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 92831
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92831(Bisanilinopyrimidine, 9d | US9249124, 47)
Affinity DataIC50:  44.9nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92831(Bisanilinopyrimidine, 9d | US9249124, 47)
Affinity DataIC50:  44.9nMpH: 7.4 T: 2°CAssay Description:Reactions were carried out at room temperature in 15 mM HEPES buffer (pH 7.4) containing 20 mM NaCl, 1 mM EGTA, 0.02% Tween 20, 10 mM MgCl2, 5% (v/v)...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92831(Bisanilinopyrimidine, 9d | US9249124, 47)
Affinity DataIC50:  180nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92831(Bisanilinopyrimidine, 9d | US9249124, 47)
Affinity DataIC50: >1.00E+4nMT: 2°CAssay Description:Specifically, MDA-MB-468 cells (American Type Culture Collection) were maintained in Dulbecco's modified Eagle's medium (DMEM) plus 10% fetus bovine ...More data for this Ligand-Target Pair
In DepthDetails US Patent