Affinity DataKd: 0.190nMAssay Description:Binding constant for PLK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.190nMAssay Description:Binding affinity to PLK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 0.810nMAssay Description:Binding constant for PLK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding constant for PLK3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding constant for RPS6KA4(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 22nMAssay Description:Binding constant for CAMKK1 kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 23nMAssay Description:Binding constant for CAMKK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRD4 expressed in Escherichia coli BL21 (DE3) cells by qPCR assayMore data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Binding affinity to human partial length BRD4 bromodomain 1 long isoform (N44 to E168 residues) expressed in bacterial expression system by competiti...More data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to recombinant human His6-TEV protease-tagged BRD4 bromodomain 1 expressed in bacteria by isothermal titration calorimetric methodMore data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to BRD4 (unknown origin) by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to His6/TEV fused recombinant human BRD4 expressed in bacteria assessed as dissociation constant by isothermal titration calorimetry...More data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to BRD4 (unknown origin) by isothermal calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 57nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRD4 expressed in Escherichia coli BL21 (DE3) cells by MST assayMore data for this Ligand-Target Pair
Affinity DataKd: 87nMAssay Description:Binding affinity to BRD4 (unknown origin) by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 97nMAssay Description:Binding constant for MYLK kinase domainMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Moffitt Cancer Center
Curated by ChEMBL
Moffitt Cancer Center
Curated by ChEMBL
Affinity DataKd: 105nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRDT expressed in Escherichia coli BL21 (DE3) cells by qPCR assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 gamma(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding constant for PIP5K2C kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 112nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRD4 expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding constant for DAPK3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for FAK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding constant for ALK kinase domainMore data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute
Curated by ChEMBL
Dana Farber Cancer Institute
Curated by ChEMBL
Affinity DataKd: 170nMAssay Description:Binding affinity to human partial length TAF1 bromodomain 2 (D1521 to D1656 residues) expressed in bacterial expression system by competitive phage d...More data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding constant for GAK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Binding constant for EGFR(L858R,T790M) kinase domainMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Moffitt Cancer Center
Curated by ChEMBL
Moffitt Cancer Center
Curated by ChEMBL
Affinity DataKd: 240nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRDT expressed in Escherichia coli BL21 (DE3) cells by MST assayMore data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:Binding constant for RPS6KA5(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding constant for PYK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:Binding constant for PRKD1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 350nMAssay Description:Binding constant for PRKD3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 360nMAssay Description:Binding constant for EGFR(T790M) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 380nMAssay Description:Binding constant for CSNK1E kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 460nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Binding constant for PRKR kinase domainMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 19(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 480nMAssay Description:Binding constant for YSK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 510nMAssay Description:Binding constant for PRKD2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 540nMAssay Description:Binding constant for DAPK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Binding constant for CLK3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Binding constant for EGFR(G719C) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 700nMAssay Description:Binding constant for RSK3(Kin.Dom.1-N-terminal) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 720nMAssay Description:Binding constant for NEK3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 770nMAssay Description:Binding constant for NIM1 kinase domainMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Moffitt Cancer Center
Curated by ChEMBL
Moffitt Cancer Center
Curated by ChEMBL
Affinity DataKd: 806nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRDT expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 850nMAssay Description:Binding constant for GRK7 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 930nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 940nMAssay Description:Binding constant for CLK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for STK33 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for EGFR(L747-E749del, A750P) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for STK16 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for JNK3 kinase domainMore data for this Ligand-Target Pair