TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to MLK1More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to PDPK1More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to TNK2More data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to JH1 catalytic domain of JAK3More data for this Ligand-Target Pair
Affinity DataKd: 57nMAssay Description:Binding affinity to PKN1More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 68nMAssay Description:Binding affinity to PDGFRBMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 68nMAssay Description:Binding affinity to FLT3More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 68nMAssay Description:Binding affinity to FLT3 catalytic domain by KinomeScan kinase binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Binding affinity to SIK2More data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity to ARK5More data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding affinity to MST2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 19(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 130nMAssay Description:Binding affinity to YSK4More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to KITMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding affinity to FGRMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding affinity to TBK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase SIK3 [59-1321](Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 230nMAssay Description:Binding affinity to QSKMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 270nMAssay Description:Binding affinity to MLK3More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 320nMAssay Description:Binding affinity to IKK-epsilonMore data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Binding affinity to MARK2More data for this Ligand-Target Pair
Affinity DataKd: 430nMAssay Description:Binding affinity to GAKMore data for this Ligand-Target Pair
Affinity DataKd: 440nMAssay Description:Binding affinity to SNARKMore data for this Ligand-Target Pair
Affinity DataKd: 460nMAssay Description:Binding affinity to LCKMore data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 490nMAssay Description:Binding affinity to MARK3More data for this Ligand-Target Pair
Affinity DataKd: 510nMAssay Description:Binding affinity to JH1 catalytic domain JAK2More data for this Ligand-Target Pair
Affinity DataKd: 550nMAssay Description:Binding affinity to GRK7More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 560nMAssay Description:Binding affinity to CSF1RMore data for this Ligand-Target Pair
Affinity DataKd: 560nMAssay Description:Binding affinity to EGFRMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TNK1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 570nMAssay Description:Binding affinity to TNK1More data for this Ligand-Target Pair
Affinity DataKd: 580nMAssay Description:Binding affinity to ZAP70More data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding affinity to BLKMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 690nMAssay Description:Binding affinity to CAMK2AMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 720nMAssay Description:Binding affinity to TAK1More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 760nMAssay Description:Binding affinity to CAMKK1More data for this Ligand-Target Pair
Affinity DataKd: 760nMAssay Description:Binding affinity to MST1More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 790nMAssay Description:Binding affinity to CAMKK2More data for this Ligand-Target Pair
Affinity DataKd: 800nMAssay Description:Binding affinity to AURKCMore data for this Ligand-Target Pair
Affinity DataKd: 850nMAssay Description:Binding affinity to PLK4More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 900nMAssay Description:Binding affinity to PDGFRAMore data for this Ligand-Target Pair
Affinity DataKd: 940nMAssay Description:Binding affinity to FYNMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 950nMAssay Description:Binding affinity to MAP3K2More data for this Ligand-Target Pair
Affinity DataKd: 960nMAssay Description:Binding affinity to HCKMore data for this Ligand-Target Pair
Affinity DataKd: 960nMAssay Description:Binding affinity to AAK1More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit delta(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to CAMK2DMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to YESMore data for this Ligand-Target Pair
TargetPhosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to PHKG1More data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding affinity to RIOK1More data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity to RIOK3More data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding affinity to PRKCDMore data for this Ligand-Target Pair