Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ki for monomerid = 121107
TargetProkineticin receptor 2(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121107(US8722896, (-)-(3R)-1-(Indolin-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  2.87nM ΔG°:  -50.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California

US Patent
LigandPNGBDBM121107(US8722896, (-)-(3R)-1-(Indolin-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  17.8nM ΔG°:  -46.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent