TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 4.64E+4nMAssay Description:Binding affinity towards sigma opioid receptor in guinea pig cerebral homogenate using [3H]DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+5nMAssay Description:Competitive inhibition of Rat liver Monoamine Oxidase B at 37 degree C (pH= 7.4)More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+5nMAssay Description:Inhibitory activity against Monoamine Oxidase B of Bovine liver in competitive inhibition assay at 25 degree C (pH=7.4)More data for this Ligand-Target Pair
Affinity DataKi: 7.60E+5nMAssay Description:In vitro inhibition of bovine monoamine oxidase B.More data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
University Of Kansas
Curated by ChEMBL
University Of Kansas
Curated by ChEMBL
Affinity DataKi: 1.38E+6nMAssay Description:In vitro binding affinity of compound towards bovine adrenal phenylethanolamine N-methyl-transferase (PNMT)More data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
University Of Kansas
Curated by ChEMBL
University Of Kansas
Curated by ChEMBL
Affinity DataKi: 1.38E+6nMAssay Description:Inhibitory activity against bovine adrenal norepinephrine N-methyl-transferase was determinedMore data for this Ligand-Target Pair