Compile Data Set for Download or QSAR
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Found 3 of ki for monomerid = 50038212
TargetMuscarinic acetylcholine receptor M1(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50038212(2-Ethyl-8-methyl-2,8-diaza-spiro[4.5]decane-1,3-di...)
Affinity DataKi:  400nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50038212(2-Ethyl-8-methyl-2,8-diaza-spiro[4.5]decane-1,3-di...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]pirenzepine from rat cortex membrane expressing muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Institute For Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50038212(2-Ethyl-8-methyl-2,8-diaza-spiro[4.5]decane-1,3-di...)
Affinity DataKi:  970nMAssay Description:Compound tested in vitro for displacement of [3H]quinuclidinyl benzilate from rat cerebellum membrane expressing muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed