Affinity DataKi: 84nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of [3H]PIA from adenosine A1 receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Inhibitory activity against adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 583nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
Affinity DataKi: 645nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Inhibition of calf intestinal adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Displacement of [3H]NECA from A2-receptor of rat striatal membranesMore data for this Ligand-Target Pair