Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidade De S£O Paulo
Curated by ChEMBL
Universidade De S£O Paulo
Curated by ChEMBL
Affinity DataKi: 43.6nMAssay Description:Binding affinity to 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Binding affinity to 5-hydroxytryptamine 1A receptor (5-HT 1A receptor, serotonin receptor) from rat cortex using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataKi: 105nMAssay Description:Binding affinity towards Serotonin transporter from rat cortex measured using [3H]-paroxetineMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Affinity of the compound at dopamine D2 receptor, (For haloperidol Ki(nM)= 1.5+/-1.2)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Affinity of the compound at 5-hydroxytryptamine 2 receptor (For ketanserin = Ki(nM)= 0.7+/-0.09)More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Affinity of the compound at 5-hydroxytryptamine 1D receptor (For sumatriptan = Ki (nM)-12+/-1.9)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Affinity of the compound at 5-hydroxytryptamine 3 receptor (For granisetron = Ki (nM)=0.3+/-0.01)More data for this Ligand-Target Pair