Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for monomerid = 50176259
TargetDelta-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]Naltrindole form human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi:  14nMAssay Description:Activity at human cloned kappa opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi:  1.60E+3nMAssay Description:Activity at human cloned mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi:  2.00E+3nMAssay Description:Opioid receptor mu 1 agonist activity with monoamine (NE, 5-HT) uptake-blocking activity in the 0.8-1 uM rangeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity towards aldosterone receptor (Mineralocorticoid receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Wroclaw Medical University

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]-dihydromorphine from mu opioid receptor in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDelta-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute

Curated by ChEMBL
LigandPNGBDBM50176259((1R,2R)-2-[(dimethylamino)methyl]-1-(3-methoxyphen...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank