Affinity DataKi: 14nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at histamine H2 receptor by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at histamine H1 receptor by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at histamine H4 receptor by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair