Affinity DataKi: 1.20E+4nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+4nMAssay Description:Concentration required for 50% inhibition of [3H]-CHA binding on rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.23E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair