Affinity DataKi: 0.940nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 259nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 279nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by using [3H]- PIA as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research
Curated by PDSP Ki Database
Leiden/Amsterdam Center For Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 1.08E+3nMAssay Description:Displacement of [3H]DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research
Curated by PDSP Ki Database
Leiden/Amsterdam Center For Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 1.19E+3nMAssay Description:Binding affinity at human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair