TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair