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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50023392'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392(CHEMBL349519 | {4-[3-(4-Amino-benzyl)-2,6-dioxo-1-...)
Affinity DataIC50:  3.40nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392(CHEMBL349519 | {4-[3-(4-Amino-benzyl)-2,6-dioxo-1-...)
Affinity DataIC50:  64nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
University Of Virginia School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392(CHEMBL349519 | {4-[3-(4-Amino-benzyl)-2,6-dioxo-1-...)
Affinity DataKd:  32nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed