Affinity DataKi: 12nMAssay Description:Binding affinity towards rat Adenosine A1 receptor using [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of specific binding of [3H]-CPX to the A1 adenosine receptor in DDT1 MF-2 (DDT) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 11.8nMAssay Description:Inhibition of [3H]-DPCPX binding to adenosine A1 receptor (AR).More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against [3H]-DPCPX binding to Adenosine A1 recepto from DDT1 MF2 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.710nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair