Affinity DataKi: 62nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor membrane (unknown origin) measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Antagonist activity at adenosine A1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Inhibition of [3H]-CHA binding to Adenosine A1 receptor in rat whole brain homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Displacement of [3H]CHA from rat cortical membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Displacement of [3H]-CHA from rat cortical membrane Adenosine A1 receptor. Parenthesis indicate 95% confidence limit.More data for this Ligand-Target Pair
Affinity DataKi: 287nMAssay Description:Binding affinity against human Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 357nMAssay Description:Binding affinity against adenosine A1 receptor in bovine cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Displacement of [3h]DPCPX from adenosine A receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of [3H]DPCPX binding to adenosine A1 receptor of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity against Adenosine A1 receptor from rat cerebral cortex was determined using [3H]-DPCPX as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of [3H]-DPCPX binding to rat cerebral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity towards Adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity against Adenosine A1 receptor from rat cerebral cortex was determined using [3H]-DPCPX as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 463nMAssay Description:Binding affinity against adenosine A1 receptor in human cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 549nMAssay Description:Displacement of [3H]-CHA from human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 549nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 549nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 549nMAssay Description:Inhibition of human recombinant adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in HEK293 cells after 60 mins by rapid filtration assayMore data for this Ligand-Target Pair