Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50375533' TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]DPCPX in rat cortical membranes in the absence of GTPMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]DPCPX in rat cortical membranes in the presence of GTP.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT1MF-2 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Agonist activity at adenosine A1 receptor assessed as inhibition of isoproterenol-stimulated cAMP accumulation in DDT1MF-2 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Affinity DataEC50: 127nMAssay Description:Effective concentration for [35S]GTP-gamma-S, binding to adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
