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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50001497'
TargetAdenosine receptor A2a(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50001497(1,7-Dimethyl-3-propyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataKi:  9.00E+3nMAssay Description:Compound was evaluated for its ability to antagonise cyclic [3H]-AMP accumulation in [3H]-adenine-labeled guinea pig cerebral cortical slices.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50001497(1,7-Dimethyl-3-propyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataKi:  2.01E+4nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50001497(1,7-Dimethyl-3-propyl-3,7-dihydro-purine-2,6-dione...)
Affinity DataEC50:  1.06E+4nMAssay Description:Relexant activity on the spontaneous tone of isolated guinea pig tracheal ring chains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed