Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50064702'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50064702(7-(3-(3,4-dimethoxyphenyl)propyl)-2-(furan-2-yl)-7...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-SCH- 58261 from human Adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50064702(7-(3-(3,4-dimethoxyphenyl)propyl)-2-(furan-2-yl)-7...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50064702(7-(3-(3,4-dimethoxyphenyl)propyl)-2-(furan-2-yl)-7...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-CGS- 21680 from rat striatal membranes Adenosine A2A receptor. Parenthesis indicate 95% confidence limits.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50064702(7-(3-(3,4-dimethoxyphenyl)propyl)-2-(furan-2-yl)-7...)
Affinity DataIC50:  20nMAssay Description:Inhibition of 1 uM NECA-stimulated cyclic AMP levels in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed