Affinity DataKi: 5nMAssay Description:Binding affinity against human adenosine A2A receptor using [3H]-CGS-21,680 (95% confidence)More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of rat recombinant adenosine receptor A2aMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]MSX-2 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatumMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to rat adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity against human post-mortem brain adenosine A2A receptor using nuclei caudati and [3H]-CGS-21,680More data for this Ligand-Target Pair