Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50125929'
TargetAdenosine receptor A2a(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50125929(2-(furan-2-yl)-8-methyl-9-(propylthio)-8H-pyrazolo...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125929(2-(furan-2-yl)-8-methyl-9-(propylthio)-8H-pyrazolo...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]SCH-58261 from human Adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125929(2-(furan-2-yl)-8-methyl-9-(propylthio)-8H-pyrazolo...)
Affinity DataIC50:  14.8nMAssay Description:Antagonist activity as inhibition of cAMP generation after agonist-modulation of human Adenosine A2A receptor with 100 nM NECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed