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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50308507'
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50308507(4-(2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)c...)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]MSX2 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50308507(4-(2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)c...)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed