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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50372571'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50372571(CHEMBL270654)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50372571(CHEMBL270654)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cells by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed