Found 17 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM21173' 
Affinity DataKi: 51nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Inhibition of [3H]ZM-241,385 binding to adenosine A2b receptorMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2b receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 63.8nMAssay Description:Binding affinity at human Adenosine A2B receptor expressed in HEK-293 cells, using [125I]-ABOPX as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement of [3H]DPCPX from human Adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement of [3H]DPCPX from human A2BAR expressed in HEK293 cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Rattus norvegicus)
National Institute Of Diabetes & Digestive & Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes & Digestive & Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 186nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Affinity DataKi: 7.32E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Displacement of PSB-12105 from recombinant human adenosine A2B receptor expressed in CHO cell membranes preincubated for 30 mins followed by PSB-1210...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Antagonist activity at human A2BR expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP production by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human A2B expressed in CHO cells assessed as stimulation of cAMP production by alphascreen assayMore data for this Ligand-Target Pair
