Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50187591'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataEC50:  335nMAssay Description:Antagonist activity at human adenosine receptor A2b expressed in CHO cell membranes assessed as inhibition of NECA-induced cAMP accumulation measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed