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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50233109'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233109(8-(1-((5-phenyl-1,2,4-oxadiazol-3-yl)methyl)-1H-py...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-ZM241385 from human A2B receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233109(8-(1-((5-phenyl-1,2,4-oxadiazol-3-yl)methyl)-1H-py...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed