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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50053923'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50053923(CHEMBL318251 | N-(9-Chloro-2-furan-2-yl-[1,2,4]tri...)
Affinity DataKi:  13.9nMAssay Description:Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50053923(CHEMBL318251 | N-(9-Chloro-2-furan-2-yl-[1,2,4]tri...)
Affinity DataKi:  13.9nMAssay Description:In vitro binding affinity at human Adenosine A3 receptor from HEK-293 cells by [125I]-AB-MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed