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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50053933'
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50053933(CHEMBL100195 | [3-(9-Chloro-2-furan-2-yl-[1,2,4]tr...)
Affinity DataKi:  32.9nMAssay Description:Binding affinity at cloned human adenosine A3 receptor expressed in HEK-293 cells was determined using [125I]-AB-MECA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50053933(CHEMBL100195 | [3-(9-Chloro-2-furan-2-yl-[1,2,4]tr...)
Affinity DataKi:  32.9nMAssay Description:In vitro binding affinity at human Adenosine A3 receptor from HEK-293 cells by [125I]-AB-MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed