Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50067098'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50067098(3,4-Dimethoxy-N-(3-pyridin-2-yl-isoquinolin-1-yl)-...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50067098(3,4-Dimethoxy-N-(3-pyridin-2-yl-isoquinolin-1-yl)-...)
Affinity DataKi:  3.10E+5nMAssay Description:Tested for antagonist activity by displacement of specific [125I]-AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed