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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50094678'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094678(2-Furan-2-yl-8-(2,4,5-tribromo-benzyl)-8H-pyrazolo...)
Affinity DataKi:  4.48E+3nMAssay Description:Displacement of [3H]-MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells; range 3650-5501More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094678(2-Furan-2-yl-8-(2,4,5-tribromo-benzyl)-8H-pyrazolo...)
Affinity DataKi:  4.48E+3nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094678(2-Furan-2-yl-8-(2,4,5-tribromo-benzyl)-8H-pyrazolo...)
Affinity DataKi:  4.47E+6nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed