Found 18 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50001885'
Affinity DataKi: 0.880nMAssay Description:Alpha-1 receptor binding studies were performed according to the methods described by Greengrass and Bremner (Eur. J. Pharmacol., 55:323-326, 1979) o...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding assay using 5-HT2A, Dopamine D2, SERT, αA1, 5-HT2C and H1 Receptors.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to alpha1 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity measured at the Alpha-1A adrenergic receptor by the inhibition of [3H]-prazosin binding to rat cortex using unlabeled WB-4101 for no...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonistic activity at alpha-1A adrenergic receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonistic activity at alpha-1A adrenergic receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) after 10 mins by calcium 5 dye based FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) after 10 mins by calcium 5 dye based FLIPR assayMore data for this Ligand-Target Pair