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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50143722'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50143722(2-{2-[4-(2,5-Dichloro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  55nMAssay Description:Binding affinity to adrenergic alpha1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50143722(2-{2-[4-(2,5-Dichloro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  55nMAssay Description:Binding affinity to adrenergic alpha1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50143722(2-{2-[4-(2,5-Dichloro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  68.3nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor through displacement of [3H]-prazosin in epididymal rat vas deferens.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed