Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50173115'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173115(CHEMBL3809840)
Affinity DataIC50:  2.20nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed