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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50392638'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50392638(CHEMBL214986)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]prazosin from human recombinant alpha1A adrenergic receptor expressed in CHO cell membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50392638(CHEMBL214986)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]prazosin from cloned human adrenergic alpha 1A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50392638(CHEMBL214986)
Affinity DataKi:  11.2nMAssay Description:Displacement of [3H]prazosin from human cloned alpha1A adrenoceptor expressed in CHO cell membranes after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed