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Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-1B adrenergic receptor' and Ligand = 'BDBM50027060'
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)
Affinity DataEC50:  63nMAssay Description:In vitro activation of human Alpha-1B receptor expressed in rat-1 fibroblasts via calcium mobilization through the Gq coupled PLC pathway as function...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)
Affinity DataEC50:  63nMAssay Description:Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)
Affinity DataEC50:  63nMAssay Description:Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)
Affinity DataEC50:  63nMAssay Description:Activation of recombinant human adrenergic, alpha-1B receptor expressed in rat-1 fibroblasts determined via calcium mobilization through Gq coupled P...Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed