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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-1D adrenergic receptor' and Ligand = 'BDBM50421641'
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421641(CHEMBL277375)
Affinity DataIC50:  40nMAssay Description:Inhibitory concentration against radioligand binding to human aAlpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50421641(CHEMBL277375)
Affinity DataEC50:  20nMAssay Description:Agonism of recombinant human alpha-1D adrenergic receptor, expressed in rat 1 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed