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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor' and Ligand = 'BDBM50196131'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Timisoara Of The Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50196131(CHEMBL217202 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  8.49nMAssay Description:Binding affinity to human cloned Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Timisoara Of The Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50196131(CHEMBL217202 | [4-(3,4-dimethylpiperazin-1-yl)phen...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed