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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Aminopeptidase N' and Ligand = 'BDBM50144922'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Aminopeptidase N


(Sus scrofa (Pig))
BDBM50144922
PNG
(CHEMBL3765787)
Show SMILES CC(C)C[C@H](NC(=O)Nc1ccc(C)cc1C)C(=O)NO
Show InChI InChI=1S/C15H23N3O3/c1-9(2)7-13(14(19)18-21)17-15(20)16-12-6-5-10(3)8-11(12)4/h5-6,8-9,13,21H,7H2,1-4H3,(H,18,19)(H2,16,17,20)/t13-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 180n/an/an/an/an/an/a



Fudan University

Curated by ChEMBL


Assay Description
Inhibition of APN in porcine kidney microsomes preincubated for 5 mins before L-leu-p-nitroanilide substrate addition for 30 mins by plate reader ana...


Eur J Med Chem 108: 21-7 (2016)


Article DOI: 10.1016/j.ejmech.2015.11.021
BindingDB Entry DOI: 10.7270/Q2ZC84RN
More data for this
Ligand-Target Pair