Affinity DataKi: 2.52E+3nMAssay Description:Displacement of [3H]-methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.76E+3nMAssay Description:Binding affinity towards testosterone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.76E+3nMAssay Description:Binding affinity for androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Binding affinity to AR (unknown origin) by FP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Displacement of [3H]methyltrienolone from androgen receptor in human LNCaP cells after 1440 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: >4.27E+4nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair