Affinity DataKi: 0.930nMAssay Description:Displacement of [125I]-Apelin-13[Glp65, Nle75, Tyr77] from YFP epitope-tagged human APJ expressed in HEK-293 cells after 1 hr by gamma counting metho...More data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Induction of HA-tagged human APJ receptor internalization expressed in HEK-293 cells after 30 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 8.60nMAssay Description:Agonist activity at human APJ receptor expressed in HEK-293 cells assessed as dissociation of G-alpha-i1 protein after 5 mins by BRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 166nMAssay Description:Agonist activity at human APJ receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair