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Found 3 Enz. Inhib. hit(s) with Target = 'Aurora kinase B' and Ligand = 'BDBM50401421'
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50401421(CHEMBL2207503)
Affinity DataIC50:  148nMAssay Description:Inhibition of Aurora B kinase-mediated Histone H3 phosphorylation at S10 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50401421(CHEMBL2207503)
Affinity DataKd:  48nMAssay Description:Binding affinity to Aurora B (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50401421(CHEMBL2207503)
Affinity DataKd:  48nMAssay Description:Binding affinity to Aurora B kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed